Molecule Details
InChIKeyQVIIMXQIBJRPFS-UHFFFAOYSA-N
Compound NameN-[4-(1-phenylpyrrolo[2,3-c]pyridin-3-yl)-2-pyridinyl]cyclopropanecarboxamide
Canonical SMILESO=C(Nc1cc(-c2cn(-c3ccccc3)c3cnccc23)ccn1)C1CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.54
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q12809 KCNH2 Homo sapiens Human PF00027 PF00520 PF13426 6.9 IC50 ChEMBL;BindingDB
Q13627 DYRK1A Homo sapiens Human PF00069 6.5 IC50 ChEMBL;BindingDB
P49841 GSK3B Homo sapiens Human PF00069 6.2 IC50 ChEMBL;BindingDB