Molecule Details
InChIKeyQVBATOUAXIHAHS-UHFFFAOYSA-N
Compound Name4-methyl-N-[5-(quinolin-8-ylcarbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-3-yl]benzamide
Canonical SMILESCc1ccc(C(=O)Nc2[nH]nc3c2CN(C(=O)c2cccc4cccnc24)C3)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.36
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 6.4 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 6.4 pIC50 TTD_MultiTarget