Molecule Details
InChIKeyQUUFDJZHDLIECK-UHFFFAOYSA-N
Compound Name5-[4-[4-(5-hydroxy-3-oxo-4H-1,4-benzoxazin-8-yl)piperazin-1-yl]butoxy]pyrazolo[1,5-a]pyridine-3-carbaldehyde
Canonical SMILESO=Cc1cnn2ccc(OCCCCN3CCN(c4ccc(O)c5c4OCC(=O)N5)CC3)cc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.66
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P14416 DRD2 Homo sapiens Human PF00001 9.1 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 8.9 Ki ChEMBL;BindingDB
P21917 DRD4 Homo sapiens Human PF00001 8.0 Ki ChEMBL;BindingDB