Molecule Details
InChIKeyQUQHXWRFOPDKOE-UHFFFAOYSA-N
Compound Name1-(6-Piperazin-1-yl-2-pyridinyl)-6-(5-propan-2-yl-3-pyridinyl)pyrazolo[4,3-c]pyridine
Canonical SMILESCC(C)c1cncc(-c2cc3c(cn2)cnn3-c2cccc(N3CCNCC3)n2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.27
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 9.9 Ki ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 9.7 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.2 Ki ChEMBL;BindingDB