Molecule Details
InChIKeyQUPOUNZWMBLXGJ-UHFFFAOYSA-N
Compound Name4-tert-butyl-N-(1-methyl-2-oxopyridin-4-yl)-2-[6-(trifluoromethyl)pyridin-3-yl]oxybenzamide
Canonical SMILESCn1ccc(NC(=O)c2ccc(C(C)(C)C)cc2Oc2ccc(C(F)(F)F)nc2)cc1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.35
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9UQD0 SCN8A Homo sapiens Human PF00520 PF24609 PF06512 PF11933 6.3 IC50 ChEMBL;BindingDB
Q9Y5Y9 SCN10A Homo sapiens Human PF00520 PF24609 PF06512 6.3 IC50 ChEMBL;BindingDB