Molecule Details
InChIKeyQUJAHTSGLDPGHW-UHFFFAOYSA-N
Canonical SMILESCOc1ccc(S(=O)(=O)N(Cc2nnn[nH]2)c2ccc(N(Cc3nnn[nH]3)S(=O)(=O)c3ccc(OC)cc3)c3ccccc23)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.81
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16236 NFE2L2 Homo sapiens Human PF03131 7.8 IC50 ChEMBL;BindingDB
Q14145 KEAP1 Homo sapiens Human PF07707 PF00651 PF01344 PF24681 7.8 IC50 ChEMBL