Molecule Details
InChIKeyQSNACFYJEZLGIS-JTQLQIEISA-N
Compound Name5-amino-2-(2,6-difluorophenyl)-N-[4-[(3S)-pyrrolidin-3-yl]oxy-3-pyridinyl]-1,3-thiazole-4-carboxamide
Canonical SMILESNc1sc(-c2c(F)cccc2F)nc1C(=O)Nc1cnccc1O[C@H]1CCNC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.0
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 9.0 IC50 ChEMBL;BindingDB
Q86V86 PIM3 Homo sapiens Human PF00069 9.0 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 9.0 IC50 ChEMBL;BindingDB