Molecule Details
InChIKeyQSMDIKOFXUXFOR-UHFFFAOYSA-N
Compound Name4-[5-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-quinoxalin-2-yl)-furan-3-yl]-benzoic acid
Canonical SMILESCC1(C)CCC(C)(C)c2nc(-c3cc(-c4ccc(C(=O)O)cc4)co3)cnc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.96
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P10826 RARB Homo sapiens Human PF00104 PF00105 8.6 IC50 ChEMBL;BindingDB
P10276 RARA Homo sapiens Human PF00104 PF00105 7.7 IC50 ChEMBL;BindingDB
P13631 RARG Homo sapiens Human PF00104 PF00105 7.6 IC50 ChEMBL;BindingDB