Molecule Details
InChIKeyQRXPIPWIGBYIFY-UHFFFAOYSA-N
Compound Name4-(5-chloro-2,4-dimethyl-1H-pyrrol-3-yl)-N-(4-fluorophenyl)pyrimidin-2-amine
Canonical SMILESCc1[nH]c(Cl)c(C)c1-c1ccnc(Nc2ccc(F)cc2)n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.44
SourceTTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 6.4 pIC50 TTD_MultiTarget
P24941 CDK2 Homo sapiens Human PF00069 6.4 pIC50 TTD_MultiTarget