Molecule Details
InChIKeyQQPVAVCRPBYZDM-UHFFFAOYSA-N
Compound Name7-Chloro-6-[1-(5-chloro-1-methylpyrazol-4-yl)sulfonylpiperidin-4-yl]-[1,2,4]triazolo[1,5-a]pyridine
Canonical SMILESCn1ncc(S(=O)(=O)N2CCC(c3cn4ncnc4cc3Cl)CC2)c1Cl
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.52
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P08912 CHRM5 Homo sapiens Human PF00001 8.1 IC50 ChEMBL
P11229 CHRM1 Homo sapiens Human PF00001 7.0 IC50 ChEMBL