Molecule Details
InChIKeyQQMKTHUGOQDEIL-UHFFFAOYSA-N
Compound NameZegocractin
Canonical SMILESCc1cccc(F)c1C(=O)Nc1cnc(-c2cc3c(cc2Cl)OC(F)(F)O3)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.48
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB16466
Drug NameCM4620
CAS Number1713240-67-5
Groups investigational
ATC Codes nan
DescriptionCM4620 (Zegocractin), is under investigation in multiple clinical trials, including NCT04195347 (pancreatitis due to asparaginase), NCT03709342 (PK/PD study in acute pancreatitis), NCT03401190 and NCT04681066 (pancreatitis and SIRS), and NCT04661540 (critical COVID-19 pneumonia).

Categories: Acids, Carbocyclic Amides Benzene Derivatives Benzoates Experimental Unapproved Treatments for COVID-19
Cross-references: CHEMBL4753998 ChemSpider: 58810276
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96D31 ORAI1 Homo sapiens Human PF07856 6.9 IC50 ChEMBL;BindingDB
Q13586 STIM1 Homo sapiens Human PF25578 PF07647 PF16533 6.5 IC50 ChEMBL
Q96SN7 ORAI2 Homo sapiens Human PF07856 6.0 IC50 ChEMBL;BindingDB