Molecule Details
InChIKeyQQFIDVOPZHXZPF-UHFFFAOYSA-N
Compound Name5-[2-Benzyl-4-(5-fluoro-2-methoxy-phenyl)-2-hydroxy-4-methyl-pentylamino]-3H-isobenzofuran-1-one
Canonical SMILESCOc1ccc(F)cc1C(C)(C)CC(O)(CNc1ccc2c(c1)COC2=O)Cc1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.97
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P06401 PGR Homo sapiens Human PF00104 PF02161 PF00105 7.1 IC50 ChEMBL;BindingDB
P04150 NR3C1 Homo sapiens Human PF02155 PF00104 PF00105 7.1 IC50 ChEMBL;BindingDB
P08235 NR3C2 Homo sapiens Human PF00104 PF00105 6.7 IC50 ChEMBL;BindingDB