Molecule Details
InChIKeyQPROYVRFSAMXGU-UHFFFAOYSA-N
Compound Name2-[[3-propan-2-yl-7-[(4-pyridin-2-ylphenyl)methylamino]-2H-pyrazolo[4,3-d]pyrimidin-5-yl]amino]butan-1-ol
Canonical SMILESCCC(CO)Nc1nc(NCc2ccc(-c3ccccn3)cc2)c2[nH]nc(C(C)C)c2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.53
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q00535 CDK5 Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB
P24864 CCNE1 Homo sapiens Human PF02984 PF00134 7.3 IC50 ChEMBL
P24941 CDK2 Homo sapiens Human PF00069 7.3 IC50 ChEMBL;BindingDB