Molecule Details
InChIKeyQPKBRNTZOUAANR-UHFFFAOYSA-N
Compound Name1-(1-cyclooctylpiperidin-4-yl)-3-(3,4-dihydro-1H-isoquinolin-2-yl)quinoxalin-2-one
Canonical SMILESO=c1c(N2CCc3ccccc3C2)nc2ccccc2n1C1CCN(C2CCCCCCC2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.57
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q5TC84 OGFRL1 Homo sapiens Human PF04664 7.4 Ki ChEMBL;BindingDB
P41145 OPRK1 Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 6.1 Ki ChEMBL;BindingDB