Molecule Details
InChIKeyQOUJDAITQNPNTN-IAGOWNOFSA-N
Compound Nametrans-(1R,2R)-N-(cyanomethyl)-2-(3,4-dihydro-1H-isoquinoline-2-carbonyl)cyclohexane-1-carboxamide
Canonical SMILESN#CCNC(=O)[C@@H]1CCCC[C@H]1C(=O)N1CCc2ccccc2C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.05
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P43235 CTSK Homo sapiens Human PF08246 PF00112 8.7 IC50 ChEMBL;BindingDB
P25774 CTSS Homo sapiens Human PF08246 PF00112 6.3 IC50 ChEMBL;BindingDB
P07858 CTSB Homo sapiens Human PF00112 PF08127 6.2 IC50 ChEMBL;BindingDB