Molecule Details
InChIKeyQOTXVDPQOVHXPX-UHFFFAOYSA-N
Compound Name4-[3-(4-Cyano-benzyl)-3H-imidazol-4-ylmethyl]-piperazine-1-carboxylic acid 2-ethoxy-benzyl ester
Canonical SMILESCCOc1ccccc1COC(=O)N1CCN(Cc2cncn2Cc2ccc(C#N)cc2)CC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL9.18
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 9.5 pIC50 TTD_MultiTarget
P53609 PGGT1B Homo sapiens Human PF00432 9.5 IC50 ChEMBL
P49356 FNTB Homo sapiens Human PF00432 8.6 IC50 ChEMBL