Molecule Details
InChIKeyQONHZAOUSLDLOE-UHFFFAOYSA-N
Compound Name2-{6-Methyl-2-[(tetrahydro-furan-2-ylmethyl)-amino]-pyrimidin-4-ylamino}-benzothiazole-6-carboxylic acid (2-chloro-6-methyl-phenyl)-amide
Canonical SMILESCc1cc(Nc2nc3ccc(C(=O)Nc4c(C)cccc4Cl)cc3s2)nc(NCC2CCCO2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.86
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P06239 LCK Homo sapiens Human PF07714 PF00017 PF00018 9.1 IC50 ChEMBL;BindingDB
P06241 FYN Homo sapiens Human PF07714 PF00017 PF00018 9.0 Ki ChEMBL;BindingDB
P12931 SRC Homo sapiens Human PF07714 PF00017 PF00018 8.5 Ki ChEMBL;BindingDB