Molecule Details
InChIKeyQNOOVTZVMOOSAW-UHFFFAOYSA-N
Compound NameEthyl (9s)-9-[5-(1h-Benzimidazol-2-Ylsulfanyl)furan-2-Yl]-8-Hydroxy-5,6,7,9-Tetrahydro-2h-Pyrrolo[3,4-B]quinoline-3-Carboxylate
Canonical SMILESCCOC(=O)c1[nH]cc2c1NC1=C(C(=O)CCC1)C2c1ccc(Sc2nc3ccccc3[nH]2)o1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.88
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 8.5 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 8.4 IC50 ChEMBL;BindingDB
P08684 CYP3A4 Homo sapiens Human PF00067 6.7 IC50 ChEMBL;BindingDB