Molecule Details
InChIKeyQNFBTXLSIOCFSM-UHFFFAOYSA-N
Compound Name3-Acetyl-4-methyl-7-[(4-pyridin-3-ylpyrimidin-2-yl)amino]chromen-2-one
Canonical SMILESCC(=O)c1c(C)c2ccc(Nc3nccc(-c4cccnc4)n3)cc2oc1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.7
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O60563 CCNT1 Homo sapiens Human PF00134 PF21797 6.7 IC50 ChEMBL;BindingDB
P50750 CDK9 Homo sapiens Human PF00069 6.7 IC50 ChEMBL
O75909 CCNK Homo sapiens Human PF00134 PF21797 6.6 IC50 ChEMBL;BindingDB