Molecule Details
InChIKeyQNAZTOHXCZPOSA-UHFFFAOYSA-N
Canonical SMILESCc1cc(OCC(=O)O)cc(C)c1Cc1ccc(O)c(C(C)C)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL9.48
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB07425
Drug NameSobetirome
CAS Number211110-63-3
Groups investigational
ATC Codes nan
Descriptionnan

Categories: Acids, Acyclic Benzene Derivatives Fatty Acids Fatty Acids, Volatile Lipids
Cross-references: BindingDB: 50115668 ChEBI: 79988 CHEMBL107400 ChemSpider: 8037944 Guide to Pharmacology: 2639 IUPHAR: 2639 C15618 PDB: B72 PubChem:9862248 PubChem:99443896 ZINC: ZINC000013475083
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P10828 THRB Homo sapiens Human PF00104 PF00105 10.0 Kd ChEMBL;BindingDB
P10827 THRA Homo sapiens Human PF00104 PF00105 9.0 Kd ChEMBL;BindingDB
DrugBank Target Actions (3)
Target Gene Target Name Action Type
P11229 CHRM1 Muscarinic acetylcholine receptor M1 agonist targets
P10828 THRB Thyroid hormone receptor beta binder targets
Q59FW3 Q59FW3 Thyroid hormone receptor alpha binder targets