Molecule Details
InChIKeyQMYPKGGBVVCXIE-UHFFFAOYSA-N
Compound Name3-[4-(4-carbamoylphenyl)-1H-pyrrolo[2,3-b]pyridin-2-yl]-N-[3-(dimethylamino)propyl]benzamide
Canonical SMILESCN(C)CCCNC(=O)c1cccc(-c2cc3c(-c4ccc(C(N)=O)cc4)ccnc3[nH]2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.0
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96RR4 CAMKK2 Homo sapiens Human PF00069 7.9 IC50 ChEMBL;BindingDB
O15111 CHUK Homo sapiens Human PF18397 PF12179 PF00069 6.9 IC50 ChEMBL;BindingDB
P45983 MAPK8 Homo sapiens Human PF00069 6.2 IC50 ChEMBL;BindingDB