Molecule Details
InChIKeyQMBXCQBKMMLGAG-UHFFFAOYSA-N
Compound Name1-[1-[3-(5-methoxy-2-methylphenoxy)-4-methylpentyl]piperidin-4-yl]-3-(1H-1,2,4-triazol-5-ylmethyl)benzimidazol-2-one
Canonical SMILESCOc1ccc(C)c(OC(CCN2CCC(n3c(=O)n(Cc4ncn[nH]4)c4ccccc43)CC2)C(C)C)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.25
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P41146 OPRL1 Homo sapiens Human PF00001 9.1 Ki ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 7.4 Ki ChEMBL;BindingDB