Molecule Details
InChIKeyQLPHOXTXAKOFMU-WBVHZDCISA-N
Canonical SMILESCNc1nc(-c2ccc3c(N)n[nH]c3c2)cc(N2C[C@@H](C(=O)NC3CCCCC3)CC[C@H]2C)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.15
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q15118 PDK1 Homo sapiens Human PF10436 PF02518 8.3 IC50 ChEMBL
O15530 PDPK1 Homo sapiens Human PF14593 PF00069 8.0 IC50 ChEMBL;BindingDB