Molecule Details
InChIKeyQLLZULWFESFQOY-OIJLLRFPSA-N
Compound NameN-(2,2-dimethylpropyl)-4-[(3R)-3-[methyl(tritritiomethyl)amino]pyrrolidin-1-yl]pyrimidin-2-amine
Canonical SMILES[3H]C([3H])([3H])N(C)[C@@H]1CCN(c2ccnc(NCC(C)(C)C)n2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.77
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9H3N8 HRH4 Homo sapiens Human PF00001 7.2 Kd ChEMBL;BindingDB
Q9Y5N1 HRH3 Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB