Molecule Details
InChIKeyQLLZULWFESFQOY-GFCCVEGCSA-N
Compound Name4-[(3R)-3-(dimethylamino)pyrrolidin-1-yl]-N-(2,2-dimethylpropyl)pyrimidin-2-amine
Canonical SMILESCN(C)[C@@H]1CCN(c2ccnc(NCC(C)(C)C)n2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.38
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9H3N8 HRH4 Homo sapiens Human PF00001 7.9 Ki ChEMBL;BindingDB
Q9Y5N1 HRH3 Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB