Molecule Details
InChIKeyQLCDJMHVAVRDAU-HNNXBMFYSA-N
Compound NameN-[(2S)-1-[(4-cyano-1-methylpiperidin-4-yl)amino]-4,4-difluoro-1-oxopentan-2-yl]-6-azaspiro[2.5]octane-6-carboxamide
Canonical SMILESCN1CCC(C#N)(NC(=O)[C@H](CC(C)(F)F)NC(=O)N2CCC3(CC2)CC3)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.22
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P25774 CTSS Homo sapiens Human PF08246 PF00112 7.6 Ki ChEMBL;BindingDB
P43235 CTSK Homo sapiens Human PF08246 PF00112 7.1 Ki ChEMBL;BindingDB
P07858 CTSB Homo sapiens Human PF00112 PF08127 7.0 Ki ChEMBL;BindingDB