Molecule Details
InChIKeyQKUXZFIUKOCULS-UHFFFAOYSA-N
Compound Name2-(3-Chloro-4-hydroxy-phenyl)-8-(1,1-dioxo-isothiazolidin-2-yl)-3-hydroxy-6-methyl-chromen-4-one
Canonical SMILESCc1cc(N2CCCS2(=O)=O)c2oc(-c3ccc(O)c(Cl)c3)c(O)c(=O)c2c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.1
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P06493 CDK1 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 6.7 pIC50 TTD_MultiTarget