Molecule Details
InChIKeyQKMUXXQVPOBBPT-VQMMKQGYSA-N
Compound Name(11E)-11-[3-[(4R,5S)-5-(4-chlorophenyl)-4-hydroxy-3,3-dimethylpiperidin-1-yl]propylidene]-5H-[1]benzoxepino[3,4-b]pyridine-9-carboxylic acid
Canonical SMILESCC1(C)CN(CC/C=C2/c3cc(C(=O)O)ccc3OCc3ncccc32)C[C@H](c2ccc(Cl)cc2)[C@H]1O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.82
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P51681 CCR5 Homo sapiens Human PF00001 9.0 Ki ChEMBL;BindingDB
P08172 CHRM2 Homo sapiens Human PF00001 8.9 Ki ChEMBL;BindingDB
P32246 CCR1 Homo sapiens Human PF00001 8.6 IC50 ChEMBL;BindingDB