Molecule Details
InChIKeyQKKGSTFAKMXWFE-UHFFFAOYSA-N
Compound NameN-(4-pyridin-4-yl-1,3-thiazol-2-yl)-2,3-dihydro-1,4-benzodioxine-3-carboxamide
Canonical SMILESO=C(Nc1nc(-c2ccncc2)cs1)C1COc2ccccc2O1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.4
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O75116 ROCK2 Homo sapiens Human PF25346 PF00069 PF08912 8.1 IC50 ChEMBL;BindingDB
Q13464 ROCK1 Homo sapiens Human PF25346 PF00069 PF08912 7.9 IC50 ChEMBL;BindingDB
P17612 PRKACA Homo sapiens Human PF00069 6.2 IC50 BindingDB