Molecule Details
InChIKeyQKJMPSJTHLLZPU-UHFFFAOYSA-N
Compound Namemethyl 4-(4-(naphthalen-2-yl)-5-oxo-3-(2-(tetrahydro-2H-pyran-4-ylamino)pyridin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-1-yl)piperidine-1-carboxylate
Canonical SMILESCOC(=O)N1CCC(n2nc(-c3ccnc(NC4CCOCC4)c3)n(-c3ccc4ccccc4c3)c2=O)CC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.1
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P53779 MAPK10 Homo sapiens Human PF00069 7.6 IC50 ChEMBL;BindingDB
P45984 MAPK9 Homo sapiens Human PF00069 7.2 IC50 ChEMBL;BindingDB
P45983 MAPK8 Homo sapiens Human PF00069 6.4 IC50 ChEMBL;BindingDB