Molecule Details
InChIKeyQJYZXCLZGZROIV-UHFFFAOYSA-N
Compound Name3-(2-amino-4-methyl-1H-benzo[d]imidazol-7-yl)-2-(1H-tetrazol-5-yl)-6-(trifluoromethyl)benzenesulfonamide
Canonical SMILESCc1ccc(-c2ccc(C(F)(F)F)c(S(N)(=O)=O)c2-c2nnn[nH]2)c2[nH]c(N)nc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.58
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 10.0 IC50 ChEMBL;BindingDB
Q5GN09 vim-1 Klebsiella pneumoniae Pathogen PF00753 9.8 IC50 BindingDB
P52699 Serratia marcescens Pathogen PF00753 8.9 IC50 BindingDB