Molecule Details
InChIKeyQJVNJCPKZBCJKQ-AREMUKBSSA-N
Canonical SMILESCN(C)CC[C@H](CSc1ccccc1)Nc1ccc(S(=O)(=O)NC(=O)c2csc(N3CCc4cccc(C(=O)Nc5nc6ccccc6s5)c4C3)n2)cc1[N+](=O)[O-]
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.68
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q07817 BCL2L1 Homo sapiens Human PF00452 PF02180 9.8 Ki ChEMBL;BindingDB
P10415 BCL2 Homo sapiens Human PF00452 PF02180 7.5 Ki ChEMBL;BindingDB