Molecule Details
InChIKeyQJRKDESSUVYBDT-UHFFFAOYSA-N
Compound Name3-[5-(Morpholin-4-ylmethyl)-1h-indol-2-yl]-1h-indazole-6-carbonitrile
Canonical SMILESN#Cc1ccc2c(-c3cc4cc(CN5CCOCC5)ccc4[nH]3)n[nH]c2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.81
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P50613 CDK7 Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB
P51946 CCNH Homo sapiens Human PF16899 PF00134 8.0 IC50 BindingDB
O14757 CHEK1 Homo sapiens Human PF00069 7.5 IC50 ChEMBL;BindingDB