Molecule Details
InChIKeyQJCVSSMPWLUMQS-UHFFFAOYSA-N
Compound Name2-[[2-[5-(tert-butylcarbamoylamino)-3-chloro-2-(2-cyclohexylethyl)-6-oxo-pyrazin-1-yl]acetyl]amino]-N-[4-(trifluoromethyl)phenyl]sulfonyl-benzamide
Canonical SMILESCC(C)(C)NC(=O)Nc1nc(Cl)c(CCC2CCCCC2)n(CC(=O)Nc2ccccc2C(=O)NS(=O)(=O)c2ccc(C(F)(F)F)cc2)c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.54
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q0ZMF1 NS3 Hepatitis C virus genotype 1b Pathogen PF02907 6.6 Ki ChEMBL;BindingDB
C1KIQ2 Hepacivirus hominis Pathogen PF02907 6.5 Ki ChEMBL