Molecule Details
InChIKeyQIYPQJHMRBXGMO-UHFFFAOYSA-N
Compound NameN-(2-(dimethylamino)ethyl)-8-isopropyl-9-oxo-8,9-dihydrothiazolo[5,4-f]quinazoline-2-carboxamidine
Canonical SMILESCC(C)n1cnc2ccc3nc(C(=N)NCCN(C)C)sc3c2c1=O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.25
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49840 GSK3A Homo sapiens Human PF00069 6.2 IC50 ChEMBL;BindingDB
P49841 GSK3B Homo sapiens Human PF00069 6.2 IC50 ChEMBL
P06493 CDK1 Homo sapiens Human PF00069 Clinical TTD_MultiTarget TTD_MultiTarget