Molecule Details
InChIKeyQISBQJCTBKCLRU-NSHDSACASA-N
Compound Name2-[[4-[(3,4-dichloro-5-methyl-1H-pyrrole-2-carbonyl)amino]-3-[(3S)-pyrrolidin-3-yl]oxybenzoyl]amino]acetic acid
Canonical SMILESCc1[nH]c(C(=O)Nc2ccc(C(=O)NCC(=O)O)cc2O[C@H]2CCNC2)c(Cl)c1Cl
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.51
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P0AES4 gyrA Escherichia coli (strain K12) Pathogen PF03989 PF00521 7.5 IC50 ChEMBL;BindingDB
P0AES6 gyrB Escherichia coli (strain K12) Pathogen PF00204 PF00986 PF21249 PF18053 PF02518 PF01751 7.5 IC50 ChEMBL