Molecule Details
InChIKeyQIDWKSGXTFVNFQ-UHFFFAOYSA-N
Compound Name7-(4-Fluorophenyl)-2-[(3-fluoro-2-pyridinyl)methyl]-8-([1,2,4]triazolo[4,3-a]pyridin-6-yl)-[1,2,4]triazolo[1,5-c]pyrimidin-5-amine
Canonical SMILESNc1nc(-c2ccc(F)cc2)c(-c2ccc3nncn3c2)c2nc(Cc3ncccc3F)nn12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.72
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P30542 ADORA1 Homo sapiens Human PF00001 8.0 IC50 ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 7.4 IC50 ChEMBL;BindingDB