Molecule Details
InChIKeyQHYSKDAWIUFROA-UHFFFAOYSA-N
Compound Name3-{6-[(2-Chlorophenyl)amino]-1H-indazol-3-YL}-5-{[4-(dimethylamino)butanoyl]amino}benzoic acid
Canonical SMILESCN(C)CCCC(=O)Nc1cc(C(=O)O)cc(-c2n[nH]c3cc(Nc4ccccc4Cl)ccc23)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.19
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P53779 MAPK10 Homo sapiens Human PF00069 8.5 IC50 ChEMBL;BindingDB
P45983 MAPK8 Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB
Q16539 MAPK14 Homo sapiens Human PF00069 6.0 IC50 ChEMBL;BindingDB