Molecule Details
InChIKeyQHXBSJRCFQZXTO-FDXDWZSASA-N
Compound Name(3S)-4-[[(2S)-1-[[(2S)-3-(1H-indol-3-yl)-1-[[[(2S)-2-[[(2S)-2-[(2-methylpropan-2-yl)oxycarbonylamino]-3-(4-sulfooxyphenyl)propanoyl]amino]hexanoyl]amino]methylamino]-1-oxopropan-2-yl]amino]-1-oxohexan-2-yl]amino]-4-oxo-3-(3-phenylpropanoylamino)butanoic acid
Canonical SMILESCCCC[C@H](NC(=O)[C@H](Cc1ccc(OS(=O)(=O)O)cc1)NC(=O)OC(C)(C)C)C(=O)NCNC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)[C@H](CCCC)NC(=O)[C@H](CC(=O)O)NC(=O)CCc1ccccc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.0
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P32238 CCKAR Homo sapiens Human PF00001 PF09193 7.0 pIC50 TTD_MultiTarget
P32239 CCKBR Homo sapiens Human PF00001 7.0 IC50 ChEMBL