Molecule Details
InChIKeyQHWXURVXTQGCOB-UHFFFAOYSA-N
Compound Name3-(6-amino-5-(1-oxo-1,2,3,4-tetrahydroisoquinolin-6-yl)pyridin-3-yl)-N-cyclopropylbenzenesulfonamide
Canonical SMILESNc1ncc(-c2cccc(S(=O)(=O)NC3CC3)c2)cc1-c1ccc2c(c1)CCNC2=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.7
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q13043 STK4 Homo sapiens Human PF11629 PF00069 6.9 IC50 ChEMBL;BindingDB
Q13188 STK3 Homo sapiens Human PF11629 PF00069 6.9 IC50 ChEMBL;BindingDB
Q9Y6E0 STK24 Homo sapiens Human PF20929 PF00069 6.3 IC50 ChEMBL;BindingDB