Molecule Details
InChIKeyQHLGSHJIJSOCMR-UHFFFAOYSA-N
Compound Name4-[1-[3-[[4-(Pyrrolidin-1-ylmethyl)benzoyl]amino]phenyl]ethylamino]quinazoline-8-carboxamide
Canonical SMILESCC(Nc1ncnc2c(C(N)=O)cccc12)c1cccc(NC(=O)c2ccc(CN3CCCC3)cc2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.9
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 8.5 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 8.4 IC50 ChEMBL;BindingDB
P23443 RPS6KB1 Homo sapiens Human PF00069 PF00433 6.8 IC50 ChEMBL;BindingDB