Molecule Details
InChIKeyQHIQMROZSSKKAH-NICAYJAGSA-N
Compound Name(R,S)-methyl 3-(3-(6-(ethylamino)-9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxy-tetrahydrofuran-2-yl)-9H-purin-2-yl)-1-hydroxyprop-2-ynyl)benzoate
Canonical SMILESCCNC(=O)[C@H]1O[C@@H](n2cnc3c(NCC)nc(C#CC(O)c4cccc(C(=O)OC)c4)nc32)[C@H](O)[C@@H]1O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.91
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P0DMS8 ADORA3 Homo sapiens Human PF00001 8.7 Ki ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB
P29274 ADORA2A Homo sapiens Human PF00001 6.8 Ki ChEMBL;BindingDB