Molecule Details
InChIKeyQHFPQUQWXGDVKK-UHFFFAOYSA-N
Compound Name2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 31
Canonical SMILESC=CCNc1nc(C)c(-c2ccnc(Nc3cccc([N+](=O)[O-])c3)n2)s1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.92
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P24941 CDK2 Homo sapiens Human PF00069 7.0 Kd ChEMBL;BindingDB
P11802 CDK4 Homo sapiens Human PF00069 6.8 pIC50 TTD_MultiTarget