Molecule Details
InChIKeyQHBZVLDXKCSSNW-VQTJNVASSA-N
Compound Name2-[6-(dimethylsulfamoyl)-1,3-benzodioxol-5-yl]-N-[(1S)-2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-phenylethyl]-N-methylacetamide
Canonical SMILESCN(C(=O)Cc1cc2c(cc1S(=O)(=O)N(C)C)OCO2)[C@H](CN1CC[C@H](O)C1)c1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.32
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P41145 OPRK1 Homo sapiens Human PF00001 9.3 Ki ChEMBL;BindingDB
P41143 OPRD1 Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB
P35372 OPRM1 Homo sapiens Human PF00001 7.5 Ki ChEMBL;BindingDB