Molecule Details
InChIKeyQGSXAJBDTYUXEY-UHFFFAOYSA-N
Compound NameN-(2-(4-(2,3-dichlorophenyl)piperazin-1-yl)ethyl)-6-methyl-2-(methylthio)pyrimidine-4-carboxamide hydrochloride
Canonical SMILESCSc1nc(C)cc(C(=O)NCCN2CCN(c3cccc(Cl)c3Cl)CC2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.8
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28223 HTR2A Homo sapiens Human PF00001 7.3 IC50 ChEMBL;BindingDB
P28335 HTR2C Homo sapiens Human PF00001 7.1 IC50 ChEMBL;BindingDB
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 6.1 IC50 ChEMBL;BindingDB