Molecule Details
InChIKeyQGNGZCPBWQOYKN-UHFFFAOYSA-N
Compound Name5-[4-(4-Bromo-phenoxy)phenyl]-5-piperazin-1-yl-pyrimidine-2,4,6-trione
Canonical SMILESO=C1NC(=O)C(c2ccc(Oc3ccc(Br)cc3)cc2)(N2CCNCC2)C(=O)N1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.5
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P14780 MMP9 Homo sapiens Human PF00040 PF00045 PF00413 8.7 IC50 ChEMBL;BindingDB
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 8.3 pIC50 TTD_MultiTarget