Molecule Details
InChIKeyQGJDHDIEZQDSIA-UHFFFAOYSA-N
Canonical SMILESCc1ccc(C(=O)Nc2ccon2)cc1NC(=O)c1cnc(NC(C)C)s1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.42
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16539 MAPK14 Homo sapiens Human PF00069 8.4 IC50 ChEMBL;BindingDB
P06239 LCK Homo sapiens Human PF07714 PF00017 PF00018 6.4 IC50 ChEMBL;BindingDB