Molecule Details
InChIKeyQGFZDGFJYXGLAW-UHFFFAOYSA-N
Compound Name3-[6-Fluoro-10-(piperidine-1-carbonyl)-1,10-diazatricyclo[6.4.1.04,13]trideca-2,4,6,8(13)-tetraen-3-yl]-4-imidazo[1,2-a]pyridin-2-ylpyrrole-2,5-dione
Canonical SMILESO=C1NC(=O)C(c2cn3c4c(cc(F)cc24)CN(C(=O)N2CCCCC2)CC3)=C1c1cn2ccccc2n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.32
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49841 GSK3B Homo sapiens Human PF00069 9.1 IC50 ChEMBL
P49840 GSK3A Homo sapiens Human PF00069 8.8 IC50 ChEMBL
Q00535 CDK5 Homo sapiens Human PF00069 7.1 IC50 ChEMBL