Molecule Details
InChIKeyQFYHJFQVDPPYCL-JOCHJYFZSA-N
Compound Name(R)-2-(Biphenyl-4-sulfonylamino)-N-hydroxy-3-(1H-indol-3-yl)-propionamide
Canonical SMILESO=C(NO)[C@@H](Cc1c[nH]c2ccccc12)NS(=O)(=O)c1ccc(-c2ccccc2)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.6
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 8.9 pIC50 TTD_MultiTarget
P14780 MMP9 Homo sapiens Human PF00040 PF00045 PF00413 8.3 IC50 ChEMBL;BindingDB