Molecule Details
InChIKeyQFVRKKGXFGGVET-UHFFFAOYSA-N
Compound Name5-(3-Chlorophenyl)-6-[[[3-(3-chlorophenyl)-4-cyanophenyl]-(3-methylimidazol-4-yl)methoxy]methyl]-1-methyl-2-oxopyridine-3-carbonitrile
Canonical SMILESCn1cncc1C(OCc1c(-c2cccc(Cl)c2)cc(C#N)c(=O)n1C)c1ccc(C#N)c(-c2cccc(Cl)c2)c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL8.34
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 9.0 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 9.0 IC50 ChEMBL
P53609 PGGT1B Homo sapiens Human PF00432 7.0 IC50 ChEMBL